Drugs to prevent Migraine

By

Beta-blockers (e.g., propranolol, metoprolol)

  • Rationale: Reduce sympathetic nervous system activity, which may play a role in migraine pathogenesis.
  • Antidepressants (e.g., amitriptyline, venlafaxine)
  • Rationale: Tricyclic antidepressants (TCAs) and serotonin-norepinephrine reuptake inhibitors (SNRIs) modulate pain pathways.
  • Antiepileptics (e.g., topiramate, valproate)
  • Rationale: Stabilize neuronal excitability, reducing cortical spreading depression.
  • CGRP antagonists (e.g., erenumab, fremanezumab)
  • Rationale: Block calcitonin gene-related peptide (CGRP), a key player in migraine pathophysiology.
  • OnabotulinumtoxinA (Botox)
  • Rationale: Inhibits neurotransmitter release at the neuromuscular junction, reducing pain transmission.
  • Calcium channel blockers (e.g., verapamil)
  • Rationale: Modulate vascular tone and neuronal excitability.
  • NSAIDs (e.g., naproxen, ibuprofen)
  • Rationale: Reduce inflammation, which may contribute to migraine.
  • Dietary supplements (e.g., riboflavin, magnesium, coenzyme Q10)
  • Rationale: May improve mitochondrial function and reduce oxidative stress.

Guidelines:

  • AHA/ASA (2021) recommend beta-blockers, TCAs, and antiepileptics as first-line options.
  • EHF (2020) suggests CGRP antagonists for patients with frequent or severe migraines.